Continuous synthesis of artemisinin-derived medicines.

نویسندگان

  • Kerry Gilmore
  • Daniel Kopetzki
  • Ju Weon Lee
  • Zoltán Horváth
  • D Tyler McQuade
  • Andreas Seidel-Morgenstern
  • Peter H Seeberger
چکیده

Described is a continuous, divergent synthesis system which is coupled to continuous purification and is capable of producing four anti-malarial APIs. The system is comprised of three linked reaction modules for photooxidation/cyclization, reduction, and derivatization. A fourth module couples the crude reaction stream with continuous purification to yield pure API.

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عنوان ژورنال:
  • Chemical communications

دوره 50 84  شماره 

صفحات  -

تاریخ انتشار 2014